CB1-IN-1

Hersteller MedChem Express
Kategorie
Typ Inhibitors
Specific against other
Menge 10mM*1mL (in DMSO)
ArtNr HY-12790-10mM
eClass 6.1 30220300
eClass 9.0 32160605
Lieferbar
CAS No.
1429239-98-4
Purity
>98%
MW
7516688
Formula
C33H31Cl2F3N6O3S2
Solubility
10 mM in DMSO
Biological Description
CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively.
IC50 value: 0.3 nM (Ki, CB1R) 21 nM (Ki, CB2R)
Target: CB1R
in vivo: CB1-IN-1 is a novel peripherally restricted cannabinoid 1 receptor antagonist with significant weight-loss efficacy in diet-induced obese mice. CB1-IN-1 has great potential to ameliorate this related metabolic syndrome.
Menge: 10mM*1mL (in DMSO)
Lieferbar: In stock
Listenpreis: 534,29 €
Preis: 534,29 €
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