ADL-5859

Hersteller MedChem Express
Kategorie Produkte / Inhibitors / Research Area / Oncology / Bladder Cancer / Testicular & Prostate Cancer
Typ Inhibitors
Specific against other
Clon N/A
Menge 100mg
ArtNr HY-13044-100mg
Eclass 6.1 30220300
Eclass 9.0 32160605
Lieferbar
Synonyms
ADL5859, ADL 5859
CAS No.
850173-95-4
Purity
>98%
MW
4289517
Formula
C24H29ClN2O3
Solubility
10 mM in DMSO
Biological Description
ADL5859 is a delta-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor kappa, u, and weak inhibitory activity at the hERG channel.
IC50 value: 0.8 nM(Ki)
Target: delta-opioid receptor
ADL-5859 (ADL5859) is an delta-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM). ADL-5859 (ADL5859) is an agonist agent that selectively stimulates the delta-opioid receptor with potential application in a wide range of inflammatory, neuropathic and acute pain conditions. In addition, Delta agonists are thought to modulate other biological processes that may manifest themselves in disease states or conditions such as overactive bladder and depression.ADL-5859 (ADL5859) is useful for inflammatory, neuropathic and acute pain conditions.
Publications
Eur J Pharmacol. 2016 Jun 15; 781:53-9.
Free  Sample
Available in quantities of 0, 5mg-1mg. Three different samples per customer per year!
Menge: 100mg
Lieferbar: In stock
Listenpreis: 1.525,36 €
Preis: 1.525,36 €
lieferbar

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