« Back
Home /
GSK2636771

GSK2636771

Item no.	V0135-5mg
Manufacturer	InvivoChem LLC
CASRN	1372540-25-4
Amount	5 mg
Quantity options	100 mg 10 mg 250 mg 25 mg 500 mg 50 mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	1372540-25-4
Available
Description	InvivoChem Cat #:V0135CAS #:1372540-25-4 Purity >=98% Description: GSK2636771 is a novel, potent, selective and orally bioavailable inhibitor of PI3Kbeta (phosphatidylinositol 3-kinase beta) with potential anticancer activity. It inhibits PI3Kbeta with a Ki of 0.89 nM and an IC50 of 5.2 nM, showing 900-fold selectivity for PI3Kbeta over p110alpha and p110gamma, and 10-fold selectivity over p110delta isoforms. Description: Description: GSK2636771 is a novel, potent, selective and orally bioavailable inhibitor of PI3Kbeta (phosphatidylinositol 3-kinase beta) with potential anticancer activity. It inhibits PI3Kbeta with a Ki of 0.89 nM and an IC50 of 5.2 nM, showing 900-fold selectivity for PI3Kbeta over p110alpha and p110gamma, and 10-fold selectivity over p110delta isoforms.inhibitor of PI3Kbeta (phosphatidylinositol 3-kinase beta) betabetaPI3Kbeta with aPI3Kbeta References:Clin Cancer Res. 2013 Jul 1; 19(13):3533-44. References:References: Related CAS: 2108806-07-9 (HCl salt); 1372540-91-4 (tris)

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

Request product datasheet

Request safety datasheet

Simple Order Order Subscription

Amount: 5 mg

available

Delivery expected until 9/4/2025

Express Delivery: Save 6 days

Compare

Add to wishlist

Get an offer