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Telotristat Etiprate (LX 1606 Hippurate)

Telotristat Etiprate (LX 1606 Hippurate)

Item no.	V0938-5mg
Manufacturer	InvivoChem LLC
CASRN	1137608-69-5
Amount	5 mg
Quantity options	100 mg 10 mg 250 mg 25 mg 500 mg 50 mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	1137608-69-5
Available
Description	InvivoChem Cat #:V0938CAS #:1137608-69-5Purity >=98% Description: Telotristat Etiprate (LX1606 etiprate; LX1032; LX-1032; LX-1606) is the a hippurate salt of telotristat ethyl, which is a prodrug of Telotristat. Telotristat ethyl is an orally bioavailable and peripheral tryptophan hydroxylase (TPH) inhibitor with potential antiserotonergic activity. Telotristat etiprate is converted to the active form, telotristat (LP-778902) Upon administration, which binds to and inhibits the activity of TPH. Telotristat etiprate is useful in controlling diarrhea associated with carcinoid syndrome. Telotristat Etiprate acts by inhibiting the enzyme tryptophan hydoxylase (TPH) and reduces serotonin production both inside and outside the GI tract without affecting brain serotonin levels. Description: References: Gut. 2014 Jun; 63(6):928-37. References: Related CAS: 1033805-28-5 (Telotristat); 1033805-22-9 (Telotristat ethyl); 1374745-52-4 (Telotristat besilate)
Molecular Weight (MW)	754.15
Formula	C27H26ClF3N6O3.C9H9NO3
CAS No.	1137608-69-5 (Telotristat etiprate);
Storage	-20C for 3 years in powder form
	-80C for 2 years in solvent
Solubility (In vitro)	DMSO: 100 mg/mL (132.6 mM)
	Water: < 1 mg/mL
	Ethanol: < 1 mg/mL
SMILES Code	O=C(OCC)[CH](N)CC1=CC=C(C2=NC(N)=NC(O[CH](C3=CC=C(Cl)C=C3N4N=C(C)C=C4)C(F)(F)F)=C2)C=C1.O=C(O)CNC(C5=CC=CC=C5)=O
Synonyms	LX1032 etiprate; LX1606 etiprate; LX 1606; LX1032 etiprate; LX 1032 etiprate; LX1606; LX 1606 Hippurate; Telotristat etiprate;

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Amount: 5 mg

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Delivery expected until 11/6/2025

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