« Back
Home /
rs-127445

rs-127445

Item no.	V0968-5mg
Manufacturer	InvivoChem LLC
CASRN	199864-87-4
Amount	5mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	199864-87-4
Available
Description	InvivoChem Cat #:V0968CAS #:199864-87-4Purity >=98% Description: RS-127445 (RS 127445; RS127445) is a novel, potent, selective, and orally bioavailable 5-HT2B receptor antagonist with important biological activity. It inhibits 5-HT2B with a pKi of 9.5 and pIC50 of 10.4, and exhibits > 1000-fold selectivity for 5-HT2B over other 5-HT receptors. Description: References: Br J Pharmacol. 1999 Jul; 127(5):1075-82; Neurogastroenterol Motil. 2010 Feb; 22(2):e69-76. References: Related CAS#: 199864-86-3 (HCl)
Molecular Weight (MW)	281.33
Formula	C17H16FN3
CAS No.	199864-87-4
Storage	-20C for 3 years in powder form
	-80C for 2 years in solvent
Solubility (In vitro)	DMSO: 56 mg/mL (199.1 mM)
	Water: < 1 mg/mL
	Ethanol: 8 mg/mL (28.4 mM)
SMILES Code	CC(C1=CC(C2=C3C=CC=CC3=C(F)C=C2)=NC(N)=N1)C
Synonyms	MT500; RS-127445; RS 127445; RS127445; MT-500; MT 500.

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

Request product datasheet

Request safety datasheet

Simple Order Order Subscription

Amount: 5mg

available

Delivery expected until 7/3/2025

Express Delivery: Save 17 days

Compare

Add to wishlist

Recommend by mail