« Back
Home /
Hexestrol (HSDB 2149)

Hexestrol (HSDB 2149)

Item no.	V1731-100mg
Manufacturer	InvivoChem LLC
CASRN	84-16-2
Amount	100 mg
Quantity options	1 g 250 mg 500 mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	84-16-2
Available
Description	InvivoChem Cat #:V1731CAS #:84-16-2Purity >=98% Description: Hexestrol (also known as HSDB 2149) is a synthetic ER agonist and also a microtubule polymerization inhibitor, which binds to ERalpha and ERbeta with EC50 of 0.07 nM and 0.175 nM, respectively. It inhibits activity of AKR1B13 with IC50 of 3.2 uM. Hexestrol inhibits the d-galactose dehydrogenase activity of thermophilus aldose 1-dehydrogenase with IC50 of 0.063 mM. Hexestrol inhibits the dehydrogenase activity of AKR1C20 towards 10 uM 4-androsten-3alpha-o1-17-one with IC50 values of 2.7 uM. References: Eur J Med Chem. 2009 Sep; 44(9):3412-24; Ann N Y Acad Sci. 2004 Dec; 1028:247-57.
Molecular Weight (MW)	270.37
Formula	C18H22O2
CAS No.	84-16-2
Storage	-20C for 3 years in powder form
	-80C for 2 years in solvent
Solubility (In vitro)	DMSO: 42 mg/mL (155.3 mM)
	Water: < 1 mg/mL
	Ethanol: 42 mg/mL (155.3 mM)
Solubility (In vivo)	30% Propylene glycol, 5% Tween 80, 65% D5W: 30 mg/mL
Synonyms	HSDB 2149; HSDB2149; HSDB-2149; Cycloestrol; Erythrohexestrol; Hexoestrol; Sinestrol

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

Request product datasheet

Request safety datasheet

Simple Order Order Subscription

Amount: 100 mg

available

Delivery expected until 10/2/2025

Express Delivery: Save 23 days

Compare

Add to wishlist

Get an offer