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DBPR108

DBPR108

Item no.	V2857-5mg
Manufacturer	InvivoChem LLC
CASRN	1186426-66-3
Amount	5 mg
Quantity options	100 mg 10 mg 250 mg 25 mg 50 mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	1186426-66-3
Available
Description	InvivoChem Cat #:V2857CAS #:1186426-66-3Purity >=98% Description: DBPR108 is a novel, potent, selective, and orally bioavailable dipeptide-derived inhibitor of DPP4 with IC50 of 15 nM; It shows no inhibition on DDP8 and DPP9. The in vivo effects of DBPR108, including inhibition of plasma DPP-IV activity and suppression of blood glucose elevation, were also demonstrated. As a potent, selective, long-acting and safe DPP-IV inhibitor, DBPR108 has the potential to be developed as a therapeutic for the treatment of type 2 diabetes mellitus. References: Bioorg Med Chem Lett. 2010 Jun 15; 20(12):3596-600.
Molecular Weight (MW)	324.39
Formula	C16H25FN4O2
CAS No.	1186426-66-3
Storage	-20C for 3 years in powder form
	-80C for 2 years in solvent
Solubility (In vitro)	DMSO: 10 mM in DMSO
	Water: < 1 mg/mL
	Ethanol:
SMILES Code	N#C[CH]1N(C(CNC(C)(C)CC(N2CCCC2)=O)=O)C[CH](F)C1
Synonyms	DBPR-108; DBPR108; DBPR 108

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 5 mg

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