Comparison

Adenosine A2A Receptor Antagonist II, SCH-58261 (2-(furan-2-yl)-7-phenethyl-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine, SCH58261, SCH 58261)

Item no. USB-217152
Manufacturer United States Biological
CASRN 160098-96-4
Amount 10 mg
Category
Type Biochemicals
Format Solid
Specific against other
Purity ≥99% (HPLC)
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Shipping condition Cool pack
Available
Manufacturer - Category
Biochemicals / Biochem-Neurochemicals
Shipping Temperature
Blue Ice
Storage Conditions
4°C
Grade
Highly Purified
Form
Supplied as an off-white solid.
EU Commodity Code
38220090
Description
A highly potent and selective antagonist of adenosine A2A receptor (Ki = 600pM). Does not affect the activity of other adenosine receptors in any significant manner (Ki = 287nM; 5uM, and > 10uM for A1, A2B, and A3 receptors, respectively). Displays neuroprotective effects in cerebral ischaemia in rats, and shown to counteract Parkinsonian-like muscle rigidity in rats.

CAS Number:
160098-96-4

Synonyms:
2-(furan-2-yl)-7-phenethyl-7H-pyrazolo[4, 3-e][1, 2, 4]triazolo[1, 5-c]pyrimidin-5-amine, SCH58261, SCH 58261

Solubility:
H2O

Molecular Formula:
C₁₈H₁₅N₇O

Primary Target:
A2A Receptor

Primary Target Ki:
600pM

Storage and Stability:
Store at 4°C under inert atmosphere. For maximum recovery of product, centrifuge the original vial prior to removing the cap.

Important Note:
This product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications without the expressed written authorization of United States Biological.

Toxicity and Hazards: 
All products should be handled by qualified personnel only, trained in laboratory procedures.
Shelf Life
1year

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 10 mg
Available: In stock
available

Compare

Add to wishlist

Get an offer

Request delivery time

Ask a technical question

Submit a bulk request

Questions about this Product?
 
Close