Comparison

Azatadine dimaleate

Item no. V1238-500mg
Manufacturer InvivoChem LLC
CASRN 3978-86-7
Amount 500 mg
Quantity options 100 mg 10 mg 1 g 250 mg 25 mg 50 mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V1238CAS #:3978-86-7Purity >=98%

Description: Azatadine dimaleate (SCH10649; SCH-10649; Idulamine; Idulian; Lergocil; Optimine; Zadine), the dimaleate salt of azatadine, is a potent histamine and cholinergic inhibitor that has been approved for treating allergic rhinitis and chronic urticaria. It inhibits histamine and cholinergic receptors with IC50s of 6.5 nM and 10 nM, respectively.

Description:

References: Agents Actions. 1974 Oct; 4(4):264-70; Clin Pharmacokinet. 1991 Nov; 21(5):372-93.

References:
Molecular Weight (MW)
522.55
Formula
C20H22N2.2C4H4O4
CAS No.
3978-86-7
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Solubility (In vitro)
DMSO: 105 mg/mL (200.9 mM)
Water: 105 mg/mL (200.9 mM)
Ethanol: < 1 mg/mL
Other info

Chemical Name: 6, 11-Dihydro-11-(1-methylpiperidin-4-ylidene)-5H-benzo[5, 6]cyclohepta[1, 2-b]pyridine dimaleate

InChi Key: SGHXFFAHXTZRQM-SPIKMXEPSA-N

InChi Code: InChI=1S/C20H22N2.2C4H4O4/c1-22-13-10-16(11-14-22)19-18-7-3-2-5-15(18)8-9-17-6-4-12-21-20(17)19; 2*5-3(6)1-2-4(7)8/h2-7, 12H, 8-11, 13-14H2, 1H3; 2*1-2H, (H, 5, 6)(H, 7, 8)/b; 2*2-1-

SMILES Code: CN1CC/C(CC1)=C2C3=CC=CC=C3CCC4=CC=CN=C4\2.O=C(O)/C=C\C(O)=O.O=C(O)/C=C\C(O)=O

Synonyms
SCH 10649; azatadine maleate; SCH10649; SCH-10649; Idulamine; Idulian; Lergocil; Optimine; Zadine

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 500 mg
Available: In stock
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