Comparison

Org 27569

Item no. V1521-50mg
Manufacturer InvivoChem LLC
CASRN 868273-06-7
Amount 50 mg
Quantity options 100 mg 10 mg 250 mg 25 mg 500 mg 5 mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V1521CAS #:868273-06-7Purity >=98%

Description: Org 27569 is a novel, potent and selective allosteric modulator of cannabinoid CB1 receptor, it induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity. Org 27569 binds to a regulatory site on the CB1 receptor target, causing a conformational change that increases the binding affinity of CB1 agonists such as CP 55, 940, while decreasing the binding affinity of CB1 antagonists or inverse agonists such as rimonabant.

Description:

References: Mol Pharmacol. 2005 Nov; 68(5):1484-95; J Biol Chem. 2012 Apr 6; 287(15):12070-82.

References:
Molecular Weight (MW)
409.95
Formula
C24H28ClN3O
CAS No.
868273-06-7
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Solubility (In vitro)
DMSO: 82 mg/mL (200.0 mM)
Water: < 1 mg/mL
Ethanol: < 1 mg/mL
SMILES
O=C(C(N1)=C(CC)C2=C1C=CC(Cl)=C2)NCCC3=CC=C(N4CCCCC4)C=C3
Synonyms
ORG27569; ORG-27569; ORG 27569

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 50 mg
Available: In stock
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