Comparison

SR9243

Item no. V1854-500mg
Manufacturer InvivoChem LLC
CASRN 1613028-81-1
Amount 500 mg
Quantity options 100 mg 10 mg 250 mg 25 mg 50 mg 5 mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V1854CAS #:1613028-81-1Purity >=98%

Description: SR9243 is a potent and selective inverse agonist of LXR. It potently reduces cancer cell viability (IC50=15–104 nM) in MTT reduction assays in prostate (PC3 and DU-145), colorectal (SW620 and HT29), and lung (HOP-62 and NCI-H23) cancer cell lines. SR9243 kills cancer cells by inhibiting lipid production and the Warburg effect. SR9243 induces cell death in multiple types of cancer and does not cause the side effects that have derailed previous attempts to target these processes.

References: Cancer Cell. 2015 Jul 13; 28(1):42-56.

Molecular Weight (MW)
626.62
Formula
C31H32BrNO4S2
CAS No.
1613028-81-1
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Solubility (In vitro)
DMSO: < 1 mg/mL
Water: < 1 mg/mL
Ethanol: N/A
Other info

Chemical Name: N-(3-bromophenethyl)-2, 4, 6-trimethyl-N-((3'-(methylsulfonyl)-[1, 1'-biphenyl]-4-yl)methyl)benzenesulfonamide

InChi Key: InChI=1S/C31H32BrNO4S2/c1-22-17-23(2)31(24(3)18-22)39(36, 37)33(16-15-25-7-5-9-29(32)19-25)21-26-11-13-27(14-12-26)28-8-6-10-30(20-28)38(4, 34)35/h5-14, 17-20H, 15-16, 21H2, 1-4H3

InChi Code: FYQFEJFTCLKXTQ-UHFFFAOYSA-N

SMILES Code: O=S(C1=C(C)C=C(C)C=C1C)(N(CCC2=CC=CC(Br)=C2)CC3=CC=C(C4=CC=CC(S(=O)(C)=O)=C4)C=C3)=O

Synonyms

SR9243; SR-9243; SR 9243

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 500 mg
Available: In stock
available

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