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GSK137647A

GSK137647A

Item no.	V2812-10mg
Manufacturer	InvivoChem LLC
CASRN	349085-82-1
Amount	10 mg
Quantity options	100 mg 250 mg 25 mg 500 mg 50 mg 5 mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Description	InvivoChem Cat #:V2812CAS #:349085-82-1Purity >=98% Description: GSK137647A, a diarylsulfonamide analog, is a novel, potent and selective agonists of the free fatty acid receptor 4 (FFA4/GPR120) with pEC50 of 6.3, 6.2, and 6.1 for human, mouse and rat FFA4, respectively. GSK137647A is selective for GPR120 over a panel of 61 other targets, including other FFARs. The free fatty acid receptor 4 (FFA4/GPR120) is a member of the G protein-coupled receptor family and is a potential 7TM (transmembrane) receptor that is involved in long-chain fatty acid-stimulated glucagon-like peptide-1 (GLP-1) secretion. FFA4 is highly expressed in the intestinal endocrine cell line STC-1 and the intestine. References: Bioorg Med Chem Lett. 2014 Jul 15; 24(14):3100-3
Molecular Weight (MW)	305.39
Formula	C??H??NO?S
CAS No.	349085-82-1
Storage	-20C for 3 years in powder form
	-80C for 2 years in solvent
Solubility (In vitro)	DMSO: >= 30 mg/mL
	Water: N/A
	Ethanol: N/A
SMILES Code	O=S(C1=CC=C(OC)C=C1)(NC2=C(C)C=C(C)C=C2C)=O
Synonyms	GSK137647; GSK-137647; GSK 137647; GSK137647A; GSK-137647A; GSK 137647A

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 10 mg

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