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gsk-269984a

gsk-269984a

Item no.	V3539-50mg
Manufacturer	InvivoChem LLC
CASRN	892664-04-9
Amount	50 mg
Quantity options	100 mg 10 mg 1 mg 250 mg 25 mg 5 mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Description	InvivoChem Cat #:V3539CAS #:892664-04-9 Purity >=98% Description: GSK-269984A is a novel and potent Prostaglandin E2 Receptor 1 (EP1) antagonist with a pIC50 of 7.9. GSK269984A was designed to overcome development issues encountered with previous EP(1) antagonists such as GW848687X and was found to display excellent activity in preclinical models of inflammatory pain. However, upon cross species pharmacokinetic profiling, GSK269984A was predicted to have suboptimal human pharmacokinetic and was thus progressed to a human microdose study. References: Bioorg Med Chem Lett. 2009 May 1; 19(9):2599-603. Related CAS#:892664-17-4 (GSK-269984B)
	Name: GSK-269984A CAS#: 892664-04-9 Chemical Formula: C20H13Cl2FNNaO3 Molecular Weight: 428.22 Elemental Analysis: C, 56.10; H, 3.06; Cl, 16.56; F, 4.44; N, 3.27; Na, 5.37; O, 11.21
Storage	-20C for 3 years in powder form
	-80C for 2 years in solvent
Technical Information	Synonym: GSK-269984A; GSK269984A; GSK 269984A Chemical Name: 2-Pyridinecarboxylic acid, 6-((5-chloro-2-((4-chloro-2-fluorophenyl)methoxy)phenyl)methyl)-, sodium salt InChi Key: ROPHIKMBWGQPQO-UHFFFAOYSA-M InChi Code: InChI=1S/C20H14Cl2FNO3.Na/c21-14-6-7-19(27-11-12-4-5-15(22)10-17(12)23)13(8-14)9-16-2-1-3-18(24-16)20(25)26; /h1-8, 10H, 9, 11H2, (H, 25, 26); /q; +1/p-1 SMILES Code: O=C(C1=NC(CC2=CC(Cl)=CC=C2OCC3=CC=C(Cl)C=C3F)=CC=C1)[O-].[Na+]

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 50 mg

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Delivery expected until 9/4/2025

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