Comparison

erteberel

Item no. V4901-250mg
Manufacturer InvivoChem LLC
CASRN 533884-09-2
Amount 250 mg
Quantity options 100 mg 10 mg 1 mg 25 mg 50 mg 5 mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V4901CAS #:533884-09-2Purity >=98%

Description: Erteberel (also known as LY500307) is a novel, potent and selective estrogen receptor beta (ERbeta) inhibitor with Ki and EC50 of 1.54 nM and 3.61 nM, respectively. It has anti-tumor activities and was developed for the treatment of benign prostatic hyperplasia. LY500307 was well tolerated in BPH patients with LUTS at doses up to 25?mg once daily for 24 weeks. The study was terminated early because of inadequate efficacy.

References: Proc Natl Acad Sci U S A. 2018 Apr 17; 115(16):E3673-E3681.; Sci Rep. 2016 Apr 29; 6:24185.


Erteberel

Name: Erteberel
CAS#: 533884-09-2
Chemical Formula: C18H18O3
Exact Mass: 282.1256
Molecular Weight: 282.339
Elemental Analysis: C, 76.57; H, 6.43; O, 17.00
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Technical Information
Synonym: LY500307; LY-500307; LY 500307
IUPAC/Chemical Name: (3aS, 4R, 9bR)-4-(4-hydroxyphenyl)-1, 2, 3, 3a, 4, 9b-hexahydrocyclopenta[c]chromen-8-ol
InChi Key: XIESSJVMWNJCGZ-VKJFTORMSA-N
InChi Code: InChI=1S/C18H18O3/c19-12-6-4-11(5-7-12)18-15-3-1-2-14(15)16-10-13(20)8-9-17(16)21-18/h4-10, 14-15, 18-20H, 1-3H2/t14-, 15+, 18+/m1/s1
SMILES Code: OC1=CC=C2C([C](CCC3)([H])[C]3([H])[CH](C4=CC=C(O)C=C4)O2)=C1

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 250 mg
Available: In stock
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