« Back
Home /
GSK-1070916

GSK-1070916

Item no.	TMO-T6129-100mg
Manufacturer	TargetMol
CASRN	942918-07-2
Amount	100 mg
Quantity options	100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mg 1 mL 200 mg 25 mg 2 mg 50 mg 5 mg
Category	Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
Purity	0,98
Smiles	CCn1cc(c(n1)-c1ccc(NC(=O)N(C)C)cc1)-c1ccnc2[nH]c(cc12)-c1cccc(CN(C)C)c1
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Alias	GSK-1070916A,GSK1070916
Shipping Condition	Cool pack
Available
Manufacturer - Targets	Tie-2\|\|\|FLT\|\|\|Apoptosis\|\|\|Aurora Kinase\|\|\|AMPK
Shipping Temperature	Cool pack
Storage Conditions	-20
Molecular Weight	507.63
Description	GSK-1070916 (GSK-1070916A) is a reversible and ATP-competitive inhibitor of Aurora B/C with IC50 of 3.5 nM/6.5 nM. It displays >100-fold selectivity against the closely related Aurora A-TPX2 complex. Phase 1.
Pathways	Apoptosis\|\|\|PI3K/Akt/mTOR signaling\|\|\|Angiogenesis\|\|\|Chromatin/Epigenetic\|\|\|Tyrosine Kinase/Adaptors\|\|\|Cell Cycle/Checkpoint

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

TMO-T6129-100mg-datasheet.pdf

Request safety datasheet

Simple Order Order Subscription

Amount: 100 mg

available

Compare

Add to wishlist

Get an offer

Request delivery time

Ask a technical question