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Casein Kinase inhibitor A86

Casein Kinase inhibitor A86

Item no.	DCC-DC11251-5mg
Manufacturer	DCChemicals
CASRN	2079069-01-3
Amount	5 mg
Quantity options	10 mg 25 mg 5 mg
Category	Neuroscience Molecular Targets for Neuroscience
Specific against	other
Smiles	FC1=CN=C(N=C1C1C=NN(C)C=1CC1CC1)NC1CCC(CC1)N
Available
Manufacturer - Applications	CKIα inhibitor A86 is a groundbreaking pan-specific inhibitor targeting Casein Kinase I (CSNK1), with a remarkable binding affinity (Kd=1-10 nM) and a specific Kd of 9.8 nM for CKIα. Beyond its primary activity, this compound also demonstrates dual inhibitory effects on the transcriptional kinases CDK7 and CDK9. Notably, it exhibits minimal to no inhibition against CDK8, CDK13, CDK11a, CDK11b, and CDK19, highlighting its selective pharmacological profile.
Molecular Weight	344, 429706335068

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 5 mg

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Delivery expected until 10/9/2025

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