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GSK778 (iBET-BD1 dihydrochloride)

GSK778 (iBET-BD1 dihydrochloride)

Item no.	DCC-DC42491-10mg
Manufacturer	DCChemicals
CASRN	2451862-42-1
Amount	10 mg
Quantity options	100 mg 10 mg
Category	Reagents & Chemicals Molecules Immunochemistry
Type	Chemicals
Applications	IC
Specific against	other
Purity	>98%
Smiles	O(C1=C(C2C(C([H])([H])[H])=NOC=2C([H])([H])[H])C([H])=C2C(=C1[H])C1=C(C([H])=N2)N=C(C([H])([H])OC([H])([H])[H])N1[C@]([H])(C([H])([H])[H])C1C([H])=C([H])C([H])=C([H])C=1[H])C([H])([H])[C@]1([H])C([H])([H])N([H])C([H])([H])C1([H])[H]
ECLASS 10.1	32160000
ECLASS 11.0	32160000
UNSPSC	12000000
Available
Manufacturer - Applications	GSK778 (iBET-BD1) is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM (BRD2 BD1), 41 nM (BRD3 BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively. GSK778 phenocopies the effects of pan-BET inhibitors in cancer models.
Molecular Weight	511, 6147

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 10 mg

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Delivery expected until 2/12/2026

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