« Back
Home /
GR-127935

GR-127935

Item no.	DCC-DC70441-1g
Manufacturer	DCChemicals
CASRN	148672-13-3
Amount	1 g
Quantity options	100 mg 1 g 250 mg
Category	In Vivo
Applications	other, IV
Specific against	other
Smiles	CC1=CC(=CC=C1C2=CC=C(C=C2)C(=O)NC3=CC(=C(C=C3)OC)N4CCN(C)CC4)C5=NOC(=N5)C
Available
Manufacturer - Applications	GR-127935 is a potent and selective 5-HT1B/1D receptor antagonist with pKi of 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptor; displays >100-fold selectivity over 5HT1A, 5-HT2A, 5-HT2C receptors and other receptor types; blocks porcine carotid vascular response to sumatriptan in vivo; orally bioavailable and centrally active.
Molecular Weight	497, 58814

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

Request product datasheet

Request safety datasheet

Simple Order Order Subscription

Amount: 1 g

available

Delivery expected until 12/11/2025

Compare

Add to wishlist

Get an offer

Request delivery time