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SBI-810 (hydrochloride)

SBI-810 (hydrochloride)

Item no.	HY-164795A-10mg
Manufacturer	MedChem Express
CASRN	2772746-58-2
Amount	10 mg
Quantity options	10 mg 5 mg
Specific against	other
Purity	99.11
Citations	[1]Lawrence Barak, et al. Compositions for and methods of treating and/or preventing pain. WO2022241186A1. 2022 November 17.\|[2]Center M N A, et al. Summer Undergraduate Research Expo[J]. 2014.
Smiles	OCCN(C)C1=CC2=C(N=C(C3(CC3)C)N=C2N4CCC(CC4)C5=C(OC)C=CC=C5)C=C1.Cl
Shipping Condition	Room temperature
Available
Manufacturer - Type	Reference compound
Manufacturer - Targets	Neurotensin Receptor
Shipping Temperature	Room Temperature
Storage Conditions	4°C (Powder, sealed storage, away from moisture)
Molecular Weight	483.05
Product Description	SBI-810 hydrochloride is a functionally selected β-arrestin-biased neurotensin receptor 1 ( NTSR1 ) allosteric modulator. SBI-810 hydrochloride modulates NTSR1 G protein signaling in a G protein-specific manner in the presence of the endogenous ligand, neurotensin (NT). SBI-810 hydrochloride fully antagonizes NT-induced activation of Gq, partially antagonizes NT-induced activation of Gi1 and is permissive of NTSR1 activation of GoA and G12 [1] [2] .
Manufacturer - Research Area	Neurological Disease
Manufacturer - Pathway	GPCR/G Protein; Neuronal Signaling
Clinical information	No Development Reported

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Amount: 10 mg

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