Comparison

RLX-33

Item no. DCC-DC60330-1g
Manufacturer DCChemicals
CASRN 2784577-71-3
Amount 1 g
Quantity options 100 mg 1 g 250 mg
Category
Type Inhibitors
Applications Blocking
Specific against other
Smiles ClC1=CC=C(C2=NOC(C3=CC=C(NC(C4CC(N(CC5=CC=CO5)C4)=O)=O)C=C3)=N2)C=C1
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Manufacturer - Applications
RLX-33 is a potent, selective and blood-brain barrier (BBB) penetrant relaxin family peptide 3 (RXFP3) antagonist, also blocks relaxin-3-induced ERK1/2 phosphorylation, with IC50 values of 2.36 μM for RXFP3, 7.82 and 13.86 μM for ERK1 and ERK2 phosphorylation, respectively. RLX-33 can block the stimulation of food intake induced by the RXFP3-selective agonist R3/I5 in rats. RLX-33 can be used for the research of metabolic syndrome[1].
Molecular Weight
462, 89

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 1 g
Available: In stock
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