Comparison

BL-1249 European Partner

Manufacturer MedChem Express
Category
Type Inhibitors
Specific against other
Amount 50 mg
Item no. HY-108596-50mg
CASRN 18200-13-0
eClass 6.1 30220300
eClass 9.0 32160605
Available
Product Description
BL-1249 is a nonsteroidal anti-inflammatory agent (NSAID) and a potassium channel activator. BL-1249 potently activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2) with EC50 values of 5.5 μM and 8.0 μM, respectively. BL-1249 extracellular application activates all TREK subfamily members but has no effect on other K2P subfamilies. BL-1249 exhibits more selective for the bladder (EC50 of 1.26 μM) than vascular tissue (EC50 of 21.0 μM)[1][2].
StorageTemperature
-20°C, 3 years (Powder)
Shipping
Blue Ice
MolecularWeight
291.35
Clinical_Information
No Development Reported
Manufacturers Research_Area
Inflammation/Immunology
Solubility
DMSO : 50 mg/mL (ultrasonic; warming; heat to 60°C)
Manufacturers Target
Potassium Channel
Pathway
Membrane Transporter/Ion Channel
Manufacturers Product type
Reference compound

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 50 mg
Available: In stock
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