ML-290

Manufacturer	MedChem Express
Category	Inhibitors
Type	Inhibitors
Specific against	other
Amount	50mg
Item no.	HY-112606-50mg
CASRN	1482500-76-4
Available
Product Description	ML-290 is a first-in-class and potent relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes, with an EC50 of 94 nM. ML290 is a biased allosteric agonist at the relaxin receptor RXFP1.
StorageTemperature	Powder -20°C 3 years, 4°C 2 years; In solvent -80°C 6 months, -20°C 1 month
Formula	C24H21F3N2O5S
References	[1].Wilson KJ, et al. Optimization of the first small-molecule relaxin/insulin-like family peptide receptor (RXFP1) agonists: Activation results in an antifibrotic gene expression profile. Eur J Med Chem. 2018 Aug 5; 156:79-92.
MolecularWeight	506.49
Research Area	Others
Solubility	DMSO : 125 mg/mL (246.80 mM; Need ultrasonic)
Target	Others
Pathway	Others

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Amount: 50mg

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Delivery expected until 4/20/2023

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