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MSC-4106

MSC-4106

Manufacturer	MedChem Express
Category	Inhibitors
Type	Inhibitors
Specific against	other
Amount	5mg
Item no.	HY-147208-5mg
CASRN	2738542-58-8
Available
Product Description	MSC-4106 is an orally active and potent inhibitor of YAP/TAZ-TEAD. MSC-4106 inhibits TEAD1 or TEAD3 auto-palmitoylation and shows inhibitory effect on NCI-H226 tumor xenograft model.
StorageTemperature	-20°C, sealed storage, away from moisture; In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Applications	Cancer-programmed cell death
Formula	C18H12F3N3O2
References	[1].Timo Heinrich, et al. Optimization of TEAD P-site binding fragment hit into in vivo active lead MSC-4106. J. Med. Chem. 2022, 65, 13, 9206–9229.
MolecularWeight	359.3
Research Area	Cancer
Solubility	DMSO : 250 mg/mL (695.80 mM; Need ultrasonic)
Target	YAP
Pathway	Stem Cell/Wnt

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Delivery expected until 4/6/2023

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