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Gabapentin

Gabapentin

Item no.	HY-A0057-5mg
Manufacturer	MedChem Express
CASRN	60142-96-3
Amount	5 mg
Quantity options	100 mg 10mM/1mL 10 mg 50 mg 5 g 5 mg
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Purity	98.0
Citations	ACS Pharmacol Transl Sci. 2023 Mar 6. Cell Rep. 2019 Dec 17;29(12):3847-3858.e5. iScience. 2023 Jun 27. J Nat Med. 2021 Sep 12. J Pain. 2019 May;20(5):577-591. Neuropharmacology. 2024 Dec 21:110276. Pharmacol Res Perspect. 2021 Oct;9(5):e00879. Sci Total Environ. 2022 Jul 10;829:154437. Eur J Drug Metab Pharmacokinet. 2022 Jun 22. [1]Fink K, et, al. Inhibition of neuronal Ca(2+) influx by gabapentin and subsequent reduction of neurotransmitter release from rat neocortical slices. Br J Pharmacol. 2000 Jun;130(4):900-6. [2]Celikyurt IK, et, al. Gabapentin, A GABA analogue, enhances cognitive performance in mice. Neurosci Lett. 2011 Apr 1;492(2):124-8. [3]Meymandi MS, et, al. Gabapentin action and interaction on the antinociceptive effect of morphine on visceral pain in mice. Eur J Anaesthesiol. 2008 Feb;25(2):129-34.
Smiles	O=C(O)CC1(CN)CCCCC1
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Shipping condition	Room temperature
Available
Manufacturer - Type	Reference compound
Manufacturer - Applications	Neuroscience-Neuromodulation
Manufacturer - Targets	Calcium Channel
Shipping Temperature	Room Temperature
Storage Conditions	Store at room temperature 3 years
Molecular Weight	171.24
Product Description	Gabapentin is a potent, orally active P/Q type Ca2+ channel blocker. Gabapentin inhibits neuronal Ca2+ influx and reduction of neurotransmitter release. Gabapentin is a GABA analog that can be used to relieve neuropathic pain[1][2][3].
Manufacturer - Research Area	Neurological Disease; Cancer
Solubility	DMSO : 1 mg/mL (ultrasonic)\|H2O : 50 mg/mL (ultrasonic)
Manufacturer - Pathway	Membrane Transporter/Ion Channel; Neuronal Signaling
Clinical information	Launched

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HY-A0057-5mg-safety-datasheet.pdf