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Pelitinib (EKB-569)

Pelitinib (EKB-569)

Item no.	S1392-10
Manufacturer	Selleckchem
CASRN	257933-82-7
Amount	10 mg
Quantity options	10 mg 100 mg 1 g 10 g 10 mM/1 ml 25 mg 5 mg 50 mg 5 g
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Smiles	CCOC1=C(C=C2C(=C1)N=CC(=C2NC3=CC(=C(C=C3)F)Cl)C#N)NC(=O)C=CCN(C)C
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	257933-82-7'
Available
Manufacturer - Targets	EGFR
Storage Conditions	2 years -80 in solvent
Information	Pelitinib (EKB-569) is a potent irreversible EGFR inhibitor with IC50 of 38.5 nM. Pelitinib (EKB-569) also slightly inhibits Src, MEK/ERK and ErbB2 with IC50s of 282 nM, 800 nM and 1255 nM, respectively. Phase2.
Pathway	Protein Tyrosine Kinase

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

S1392-10-datasheet.pdf

S1392-10-safety-datasheet.pdf