Comparison

Formoterol Hemifumarate European Partner

Manufacturer Selleckchem
Category
Type Inhibitors
Specific against other
Amount 10 mg
Item no. S2020-10
CASRN 43229-80-7
eClass 6.1 30220300
eClass 9.0 32160605
Available
Chemical Name
N-(2-hydroxy-5-((S)-1-hydroxy-2-((S)-1-(4-methoxyphenyl)propan-2-ylamino)ethyl)phenyl)formamide hemifumaric acid
Description
Formoterol hemifumarate is a potent, selective and long-acting 2-adrenoceptor agonist to 2 and 1 receptors with pKd of 8.12 and 5.58, respectively. Formoterol hemifumarate reveals 330-fold selectivity for2 over 1 receptors. Formoterol hemifumarate potently relaxes guinea pig trachea (pD2 = 9.29), and is longer-acting and 100-fold more potent than salbutamol. [1] Formoterol hemifumarate works like other 2-agonists, causing bronchodilation by relaxing the smooth muscle in the airway so as to treat the exacerbation of asthma. The long duration of formoterol action occurs because the formoterol molecules initially diffuse into the plasma membrane of the lung cells, and then are slowly released back outside, where they can come into contact with 2 adrenergic receptors. [2]
Molecular Weight (MW)
402, 4
Picture ChemicalStructure Description
Formoterol hemifumarate Chemical Structure
Solubility (25C)
DMSO 98 mg/mL, Water <1 mg/mL, Ethanol <1 mg/mL
Storage
2 years -20CPowder, 2 weeks4Cin DMSO, 2 months-80Cin DMSO

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 10 mg
Available: In stock
available

Delivery expected until 4/11/2024 

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