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PF-3716556

PF-3716556

Item no.	S2222-10
Manufacturer	Selleckchem
CASRN	928774-43-0
Amount	10 mg
Quantity options	10 mg 1 g 10 g 50 mg 5 g
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Smiles	CC1=C2C(CCOC2=CC=C1)NC3=CC(=CN4C3=NC(=C4)C)C(=O)N(C)CCO
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	Proton Pump
Similar products	PF
Available
Storage Conditions	2 years -80 in solvent
Molecular Weight	394, 47
Information	PF 3716556 is a potent and selective P-CAB (potassium-competitive acid blocker), with pIC50 of 6.026 and 7.095 for the inhibition of porcine H+, K+-ATPase activity in ion-leaky and ion-tight assay, respectively, inhibits gastric acid secretion, displays no activity at Na+, K+-ATPase, used for the treatment of gastroesophageal reflux disease.
Chemical Name	(R)-N-(2-hydroxyethyl)-N, 2-dimethyl-8-(5-methyl-3, 4-dihydro-2H-chromen-4-ylamino)H-imidazo[1, 2-a]pyridine-6-carboxamide

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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S2222-10-datasheet.pdf

S2222-10-safety-datasheet.pdf