Comparison

Rupatadine European Partner

Item no. TMO-T36618-100mg
Manufacturer TargetMol
CASRN 158876-82-5
Amount 100 mg
Quantity options 100 mg 10 mg 25 mg 500 mg 50 mg 5 mg
Category
Type Inhibitors
Specific against other
Purity 0,98
Formula C26H26ClN3
Smiles ClC=1C=CC2=C(C1)CCC=3C=CC=NC3C2=C4CCN(CC=5C=NC=C(C5)C)CC4
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Alias UR-12592,UR12592
Shipping Condition Cool pack
Available
Manufacturer - Targets
PAFR|||Histamine Receptor
Shipping Temperature
Cool pack
Storage Conditions
-20
Molecular Weight
415.96
Description
Rupatadine (UR-12592, rupatadine) is a potent and orally available dual antagonist of PAF and histamine H1 receptors with Ki values of 0.55 μM and 0.1 μM, respectively, which provides relief of allergic symptoms and anti-inflammatory properties, and is used in allergic rhinitis and chronic urticaria.
Pathways
Neuroscience|||Immunology/Inflammation|||GPCR/G Protein
Bioactivity
Rupatadine (UR-12592) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM(rabbit platelet membranes/guinea pig cerebellum membranes).

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 100 mg
Available: In stock
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