Comparison

BMS-536924 European Partner

Item no. TMO-T6419-200mg
Manufacturer TargetMol
CASRN 468740-43-4
Amount 200 mg
Quantity options 100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mg 1 mL 200 mg 25 mg 2 mg 500 mg 50 mg 5 mg
Category
Type Inhibitors
Specific against other
Purity 0,9919
Formula C25H26ClN5O3
Smiles Cc1cc(cc2nc([nH]c12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCOCC1
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Alias CS-0117,BMS 536924
Shipping Condition Cool pack
Available
Manufacturer - Targets
MEK|||FAK|||Apoptosis|||Src|||IGF-1R
Shipping Temperature
Cool pack
Storage Conditions
-20
Molecular Weight
479.96
Description
BMS-536924 (BMS 536924) is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for Akt1, MAPK1/2.
Pathways
Apoptosis|||Angiogenesis|||MAPK|||Cytoskeletal Signaling|||Tyrosine Kinase/Adaptors
Bioactivity
BMS-536924 is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for Akt1, MAPK1/2.

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 200 mg
Available: In stock
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