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5-HT4 antagonist 1

5-HT4 antagonist 1

Item no.	HY-100170-1mg
Manufacturer	MedChem Express
CASRN	261766-73-8
Amount	1 mg
Quantity options	100 mg 10 mM/1 mL 10 mg 1 ea 1 mg 25 mg 50 mg 5 mg
Category	Neuroscience Molecular Targets for Neuroscience Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Purity	98.95
Citations	[1]Clark RD, et al. Identification of a 5-HT4 receptor antagonist clinical candidate through side-chain modification. Bioorg Med Chem Lett. 2005 Mar 15;15(6):1697-700.
Smiles	O=C(C1=C2OCCOC2=CC=C1)NCC3CCN(CCCS(=O)(N4CCN(C)CC4)=O)CC3
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	261766-73-8
Shipping Condition	Room temperature
Available
Manufacturer - Type	Reference compound
Manufacturer - Applications	Neuroscience-Neuromodulation
Manufacturer - Targets	5-HT Receptor
Shipping Temperature	Room Temperature
Storage Conditions	-20°C, 3 years; 4°C, 2 years (Powder)
Molecular Weight	480.62
Product Description	5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6.
Manufacturer - Research Area	Neurological Disease
Solubility	DMSO: 20 mg/mL (ultrasonic; warming; adjust pH to 3 with HCl; heat to 60°C)
Manufacturer - Pathway	GPCR/G Protein; Neuronal Signaling
Isoform	Apolipoprotein D
Clinical information	No Development Reported

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HY-100170-1mg-safety-datasheet.pdf