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Gefapixant

Gefapixant

Manufacturer	MedChem Express
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Amount	10 mg
Item no.	HY-101588-10mg
Targets	P2X Receptor
CASRN	1015787-98-0
eClass 6.1	30220300
eClass 9.0	32160605
Available
Product Description	Gefapixant is an orally active and potent purinergic P2X3 receptor (P2X3R) antagonist, with IC50 values of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. Gefapixant can be used for the research of chronic cough and knee osteoarthritis[1][2][3].
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	COVID-19-anti-virus
MolecularWeight	353.40
Clinical_Information	Launched
Manufacturers Research_Area	Inflammation/Immunology
Solubility	DMSO : 5 mg/mL (ultrasonic; adjust pH to 5-6 with HCl)
Manufacturers Target	P2X Receptor
Isoform	P2X3 Receptor
Pathway	Membrane Transporter/Ion Channel
Manufacturers Product type	Reference compound

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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HY-101588-10mg-safety-datasheet.pdf