Comparison

Fasudil (Hydrochloride) European Partner

Manufacturer MedChem Express
Category
Type Inhibitors
Specific against other
Clone N/A
Amount 500 mg
Quantity options 10 mM/1mL 1 g 200 mg 500 mg 5g
Item no. HY-10341-500mg
Targets ROCK; Calcium Channel; Autophagy; PKA; PKC; HIV
CASRN 105628-07-7
eClass 6.1 30220300
eClass 9.0 32160605
Available
Product Description
Fasudil (HA-1077; AT877) Hydrochloride is a nonspecific RhoA/ROCK inhibitor and also has inhibitory effect on protein kinases, with an Ki of 0.33 μM for ROCK1, IC50s of 0.158 μM and 4.58 μM, 12.30 μM, 1.650 μM for ROCK2 and PKA, PKC, PKG, respectively. Fasudil Hydrochloride is also a potent Ca2+ channel antagonist and vasodilator[1][2][3].
StorageTemperature
4°C (Powder, sealed storage, away from moisture)
Shipping
Room Temperature
Manufacturers Applications
Cancer-Kinase/protease
MolecularWeight
327.83
Clinical_Information
Launched
Manufacturers Research_Area
Cancer
Solubility
DMSO : ≥ 31 mg/mL|H2O : 55 mg/mL (ultrasonic)
Manufacturers Target
Autophagy; Calcium Channel; HIV; PKA; PKC; ROCK
Isoform
PKA; PKC; ROCK1; ROCK2
Manufacturers Pathway
Anti-infection; Autophagy; Cell Cycle/DNA Damage; Cytoskeleton; Epigenetics; Membrane Transporter/Ion Channel; Neuronal Signaling; Stem Cell/Wnt; TGF-beta/Smad
Manufacturers Product type
Reference compound

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 500 mg
Available: In stock
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