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GLP-1R Antagonist 1

GLP-1R Antagonist 1

Item no.	CS-0020879-25mg
Manufacturer	ChemScene
Amount	25mg
Category	Metabolism Diabetes Glucose Homeostasis Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Alias	488097-06-9
Similar products	488097-06-9
Available
CAS	488097-06-9
Purity	>98%
MWt	440.73
Formula	C16H11ClF6N4O2
Solubility	10 mM in DMSO
Clinical Information	No Development Reported
Pathway	GPCR/G Protein
Target	Glucagon Receptor
Biological Activity	GLP-1R Antagonist 1 (compound 5d) is an orally active, CNS penetrant and non-competitive antagonist of glucagon-like peptide 1 receptor (GLP-1R), with an IC₅₀ of 650 nM^[1]. IC50 & Target: IC50: 650 nM (GLP-1R)^[1].
Research Area	Metabolic Disease

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 25mg

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Delivery expected until 10/2/2025

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