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3-Phenyltoxoflavin

3-Phenyltoxoflavin

Item no.	CS-0094927-10mg
Manufacturer	ChemScene
Amount	10mg
Category	Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Alias	32502-63-9
Similar products	32502-63-9
Available
CAS	32502-63-9
Purity	>98%
MWt	269.26
Formula	C13H11N5O2
Solubility	DMSO : 7.14 mg/mL (26.52 mM; Need ultrasonic)
Clinical Information	No Development Reported
Pathway	Metabolic Enzyme/Protease; Cell Cycle/DNA Damage
Target	HSP; HSP
Biological Activity	3-Phenyltoxoflavin, a derivative of Toxoflavin, is an Hsp90 inhibitor, with a Kd of 585 nM for the interaction of Hsp90-TPR2A. 3-Phenyltoxoflavin has anti-cancer activity. In Vitro: 3-Phenyltoxoflavin (1 nM-100 uM; 4 d) inhibits BT474 cells proliferation in a concentration-dependent manner, with an IC50 of 690 nM. 3-Phenyltoxoflavin (0.56 nM-100 uM; 2 h) competes with biotinylated Hsp90 peptide for its binding to TPR2A in a dose-dependent manner.

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Amount: 10mg

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