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Glucocorticoid receptor agonist-1

Glucocorticoid receptor agonist-1

Item no.	CS-0145653-5mg
Manufacturer	ChemScene
Amount	5mg
Category	Oncology By Cell Type Carcinoma Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Alias	2166375-82-0
Similar products	2166375-82-0
Available
CAS	2166375-82-0
Purity	>98%
MWt	569.69
Formula	C35H39NO6
Solubility	10 mM in DMSO
Clinical Information	No Development Reported
Pathway	GPCR/G Protein
Target	Glucocorticoid Receptor
Biological Activity	Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC₅₀ of 2.8 nM extracted from patent WO2017210471A1, compound 41^[1]. IC50 & Target: IC50: 2.8 nM (Glucocorticoid receptor)^[1] In Vitro: Glucocorticoid receptor agonist immunoconjugates are useful for treating autoimmune diseases such as, but not limited to, rheumatoid arthritis, juvenile idiopathic arthritis, psoriatic arthritis, ankylosing spondylitis, adult Crohn's disease, pediatric Crohn's disease, ulcerative colitis, plaque psoriasis, hidradenitis suppurativa, uveitis, Behcets disease, a spondyloarthropathy, or psoriasis^[1].
Research Area	Inflammation/Immunology

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 5mg

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