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PD 151746

PD 151746

Item no.	CS-5401-100mg
Manufacturer	ChemScene
Amount	100mg
Category	Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Similar products	179461-52-0
Available
CAS	179461-52-0
Purity	>98%
Formula	C11H8FNO2S
MWt	237.25
Solubility	DMSO : >= 37 mg/mL (155.95 mM)
Clinical Information	No Development Reported
Pathway	Metabolic Enzyme/Protease
Target	Proteasome
Biological Activity	PD151746 is a calpain inhibitor, shows a 20-fold selectivity for u-calpain (Ki = 0.26 +/- 0.03 uM) over m-calpain (Ki = 5.33 +/- 0.77 uM). IC50 value: 0.26 +/- 0.03 uM (Ki, for u-calpain), 5.33 +/- 0.77 uM (Ki, for m-calpain) [1] Target: calpain in vitro: The u-calpain inhibitor PD 151746 decreases oxLDL-induced cytotoxicity. [2]

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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