Comparison

BRD9539

Item no. CS-5862-50mg
Manufacturer ChemScene
Amount 50mg
Category
Type Molecules
Specific against other
ECLASS 10.1 32169090
ECLASS 11.0 32169090
UNSPSC 12000000
Similar products 1374601-41-8
Available
CAS
1374601-41-8
Purity
>98%
Formula
C24H21N3O3
MWt
399.44
Solubility
DMSO : >= 35 mg/mL (87.62 mM)
Clinical Information
No Development Reported
Pathway
Epigenetics
Target
Histone Methyltransferase
Biological Activity
BRD9539 inhibits G9a activity with an IC50 of 6.3 uM, inhibits PRC2 activity with a similar IC50. target: G9a, PRC2; IC50: 6.3 uM ( G9a ), 6.3 uM ( PRC2 ); BRD9539 is a more potent biochemical inhibitor than its methyl-ester analogue BRD4770, with 20% remaining G9a activity compared to 45% of BRD4770 at screening concentration.

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 50mg
Available: In stock
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