Comparison

CCG-50014

Item no. DCC-DC22819-1g
Manufacturer DCChemicals
CASRN 883050-24-6
Amount 1 g
Quantity options 100 mg 1 g 250 mg
Category
Type Inhibitors
Applications IC, other
Specific against other
Purity >98%
Smiles FC1C=CC(CN2C(=O)SN(C3C=CC(C)=CC=3)C2=O)=CC=1
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Alias CCG50014,CCG 50014
Similar products 883050-24-6
Available
Manufacturer - Applications
CCG-50014 is the most potent against the regulator of G-protein signaling protein type 4 (RGS4) (IC50 =30 nM) and is >20-fold selective for RGS4 over other RGS proteins. CCG-50014 binds covalently to the RGS, forming an adduct on two cysteine residues located in an allosteric regulatory site. CCG50014, reduces nociceptive responses and enhances opioid-mediated analgesic effects in the mouse formalin test.
Molecular Weight
316, 35
Chemical name
4-[(4-Fluorophenyl)methyl]-2-(4-methylphenyl)-1, 2, 4-thiadiazolidine-3, 5-dione

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 1 g
Available: In stock
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