« Back
Home /
GSK046 (iBET-BD2)

GSK046 (iBET-BD2)

Item no.	DCC-DC39702-1g
Manufacturer	DCChemicals
CASRN	2474876-09-8
Amount	1 g
Quantity options	100 mg 1 g 250 mg
Category	Oncology By Cell Type Melanoma Reagents & Chemicals Molecules
Type	Inhibitors
Specific against	other
Smiles	O=C(N[C@H]1CC[C@H](O)CC1)C2=CC(O[C@H](C3=CC=CC=C3)C)=C(NC(C)=O)C(F)=C2
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	2474876-09-8
Similar products	2474876-09-8
Available
Manufacturer - Applications	GSK046 (iBET-BD2) is a potent, selective and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively. GSK046 has immunomodulatory activity.
Molecular Weight	414, 47

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

Request product datasheet

Request safety datasheet

Simple Order Order Subscription

Amount: 1 g

available

Delivery expected until 8/21/2025

Express Delivery: Save 3 days

Compare

Add to wishlist

Get an offer