Comparison

Gefapixant European Partner

Item no. TMO-T5099-2mg
Manufacturer TargetMol
CASRN 1015787-98-0
Amount 2 mg
Quantity options 100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mL 1 mg 200 mg 25 mg 2 mg 50 mg 5 mg
Category
Type Molecules
Format Powder
Specific against other
Purity 0,9926
Smiles COc1cc(C(C)C)c(Oc2cnc(N)nc2N)cc1S(N)(=O)=O
ECLASS 10.1 32169090
ECLASS 11.0 32169090
UNSPSC 12000000
Alias RO 4926219,AF219,MK-7264
Shipping Condition Cool pack
Available
Manufacturer - Targets
P2X Receptor
Shipping Temperature
Cool pack
Storage Conditions
-20
Molecular Weight
353.4
Description
Gefapixant (AF219) is a P2X3 receptor (P2X3R) antagonist with IC50 of ~30 nM at recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors.
Pathways
Membrane transporter/Ion channel|||Neuroscience

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 2 mg
Available: In stock
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