Comparison

azasetron-hcl-y-25130

Manufacturer InvivoChem LLC
Category
Type Biochemicals
Specific against other
Amount 1g
Item no. V1000-1g
CASRN 123040-16-4
eClass 6.1 32160405
eClass 9.0 32160490
Available
Description
InvivoChem Cat #:V1000CAS #:123040-16-4Purity >=98%

Description: Azasetron HCl (formerly Y 25130 HCl; Y-25130; Y25130), an approved antiemetic drug, is a potent and selective antagonist of 5-HT3 receptor with an IC50 of 0.33 nM. It is an antiemetic agent primarily used for the treatment of cancer chemotherapy-induced nausea and vomiting.

Description:

References: Jpn J Pharmacol. 1993 Nov; 63(3):377-83; Eur J Pharmacol. 1991 Apr 24; 196(3):299-305.

References:
Molecular Weight (MW)
386.27
Formula
C17H20ClN3O3.HCl
CAS No.
123040-16-4
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Solubility (In vitro)
DMSO: < 1 mg/mL
Water: 3 mg/mL (7.8 mM)
Ethanol: < 1 mg/mL
Other info

Chemical Name: 2H-1, 4-Benzoxazine-8-carboxamide, 3, 4-dihydro-N-1-azabicyclo(2.2.2)oct-3-yl-6-chloro-4-methyl-3-oxo-, monohydrochloride

InChi Key: DBMKBKPJYAHLQP-BTQNPOSSSA-N

InChi Code: InChI=1S/C17H20ClN3O3.ClH/c1-20-14-7-11(18)6-12(16(14)24-9-15(20)22)17(23)19-13-8-21-4-2-10(13)3-5-21; /h6-7, 10, 13H, 2-5, 8-9H2, 1H3, (H, 19, 23); 1H/t13-; /m1./s1

SMILES Code: c1(cc(C(N[CH]2CN3CCC2CC3)=O)c2c(c1)N(C)C(=O)CO2)Cl.Cl

Synonyms
Y 25130 HCl; Y-25130; Y25130

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 1g
Available: In stock
available

Delivery expected until 6/6/2024 

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