Comparison

Asenapine maleate (Org 5222 maleate)

Item no. V1097-25mg
Manufacturer InvivoChem LLC
CASRN 85650-56-2
Amount 25 mg
Quantity options 100 mg 1 g 250 mg 2 g 500 mg 50 mg 5 g
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Alias 85650-56-2
Available
Description
InvivoChem Cat #:V1097CAS #:85650-56-2Purity >=98%

Description: Asenapine maleate (Org5222; Org-5222; HSDB-8061; HSDB8061; Saphris and Sycrest), an atypical antipsychotic, is a potent and high-affinity antagonist of serotonin, norepinephrine, dopamine and histamine receptors. Asenapine has been approved as an atypical antipsychotic for the treatment of schizophrenia and acute mania associated with bipolar disorders. Preliminary data indicate that it has minimal anticholinergic and cardiovascular side effects, as well as minimal weight gain. It was approved by FDA in August 2009.

Description:

References: J Psychopharmacol. 2009 Jan; 23(1):65-73; Psychopharmacology (Berl). 2008 Feb; 196(3):417-29.

References:

Related CAS #: 85650-56-2 (maleate); 65576-45-6 (free); 1412458-61-7 (HCl)

Molecular Weight (MW)
401.84
Formula
C17H16ClNO.C4H4O4
CAS No.
85650-56-2
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Solubility (In vitro)
DMSO: 80 mg/mL (199.1 mM)
Water: < 1 mg/mL
Ethanol: < 1 mg/mL
Other info

Chemical Name: (3aS, 12bS)-5-chloro-2-methyl-2, 3, 3a, 12b-tetrahydro-1H-dibenzo[2, 3:6, 7]oxepino[4, 5-c]pyrrole maleate

InChi Key: GMDCDXMAFMEDAG-CHHFXETESA-N

InChi Code: InChI=1S/C17H16ClNO.C4H4O4/c1-19-9-14-12-4-2-3-5-16(12)20-17-7-6-11(18)8-13(17)15(14)10-19; 5-3(6)1-2-4(7)8/h2-8, 14-15H, 9-10H2, 1H3; 1-2H, (H, 5, 6)(H, 7, 8)/b; 2-1-/t14-, 15-; /m1./s1

SMILES Code: CN1C[C](C2=CC=CC=C2OC3=CC=C(Cl)C=C34)([H])[C]4([H])C1.O=C(O)/C=C\C(O)=O

Synonyms
Org 5222; HSDB 8061; Org 5222; HSDB 8061; Org5222; Org-5222; HSDB-8061; HSDB8061; Asenapine; Asenapine maleate; trade names Saphris and Sycrest.

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 25 mg
Available: In stock
available

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