Comparison

Otenabant (CP-945598)

Item no. V26985-10mg
Manufacturer InvivoChem LLC
CASRN 686344-29-6
Amount 10 mg
Quantity options 100 mg 250 mg 25 mg 500 mg 50 mg 5 mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V26985CAS #:686344-29-6Purity >=98%

Description:Otenabant free base (also known as CP-945, 598) is a novel, potent and highlyselective cannabinoid receptor CB1 antagonist with Ki of 0.7 nM, itexhibits > 10, 000-fold greater selectivity against human CB2 receptor.Otenabant is a approved drug developed by Pfizer for the treatment ofobesity, but development for this drug has been discontinued due to theproblems seen during clinical use of the similar drug rimonabant.

References: J Med Chem. 2009 Jan 22; 52(2):234-7; Biochem Biophys Res Commun. 2010 Apr 2; 394(2):366-71.

Related CAS#: 686344-29-6 (free base); 86347-12-6 (HCl)

Description:Otenabant free base (also known as CP-945, 598) is a novel, potent and highlyselective cannabinoid receptor CB1 antagonist with Ki of 0.7 nM, itexhibits > 10, 000-fold greater selectivity against human CB2 receptor.Otenabant is a approved drug developed by Pfizer for the treatment ofobesity, but development for this drug has been discontinued due to theproblems seen during clinical use of the similar drug rimonabant.

Description:

References: J Med Chem. 2009 Jan 22; 52(2):234-7; Biochem Biophys Res Commun. 2010 Apr 2; 394(2):366-71.

References:

Related CAS#: 686344-29-6 (free base); 86347-12-6 (HCl)

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 10 mg
Available: In stock
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