Comparison

L-368,899 hydrochloride European Partner

Item no. TMO-T11794-500mg
Manufacturer TargetMol
CASRN 160312-62-9
Amount 500 mg
Quantity options 100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mg 1 mL 200 mg 25 mg 2 mg 500 mg 50 mg 5 mg
Category
Type Chemicals
Specific against other
Formula C26H43ClN4O5S2
Smiles Cl.[H][C@@]12CC[C@](CS(=O)(=O)N3CCN(CC3)c3ccccc3C)(C(C1)NC(=O)[C@H](N)CCS(C)(=O)=O)C2(C)C
ECLASS 10.1 32160000
ECLASS 11.0 32160000
UNSPSC 12000000
Alias L-368899 hydrochloride,L-368,899 HCl
Shipping Condition Cool pack
Available
Manufacturer - Targets
OX Receptor
Shipping Temperature
Cool pack
Storage Conditions
-20
Molecular Weight
591.23
Description
L-368, 899 hydrochloride is an orally available and selective nonpeptide oxytocin receptor (OXTR) antagonist for the prevention of preterm labor.L-368, 899 hydrochloride prevents oxytocin-induced anti-anomalous pain and anti-nausea, and may be useful for the study of depression.
Pathways
Neuroscience|||GPCR/G Protein
Bioactivity
L-368, 899 hydrochloride, used as a tocolytic agent, is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor, respectively.

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 500 mg
Available: In stock
available

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