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Telcagepant

Telcagepant

Item no.	TMO-T16093-500mg
Manufacturer	TargetMol
CASRN	781649-09-0
Amount	500 mg
Quantity options	100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mg 1 mL 200 mg 2 mg 500 mg 50 mg 5 mg
Category	Reagents & Chemicals Biochemicals
Type	Chemicals
Specific against	other
Formula	C26H27F5N6O3
Smiles	O=C1N(C=2C(N1)=NC=CC2)C3CCN(C(N[C@H]4C(=O)N(CC(F)(F)F)C[C@@H](CC4)C5=C(F)C(F)=CC=C5)=O)CC3
ECLASS 10.1	32160000
ECLASS 11.0	32160000
UNSPSC	12000000
Alias	MK-0974,MK0974
Shipping Condition	Cool pack
Available
Manufacturer - Targets	CGRP Receptor
Storage Conditions	-20
Molecular Weight	566.52
Description	Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors and reduces neurotransmission in the central nervous system and is used in the study of migraines and for pain relief.
Pathways	Neuroscience\|\|\|GPCR/G Protein
Bioactivity	Telcagepant is an orally active antagonist of calcitonin gene-related peptide (CGRP) receptor (Kis: 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively).

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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