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DA-3003-1

DA-3003-1

Item no.	TMO-T16357-1ml
Manufacturer	TargetMol
CASRN	383907-43-5
Amount	1 mL
Quantity options	100 mg 1 mL x 10 mM (in DMSO) 1 mL x 10 mM (in DMSO) 10 mg 1 mg 1 mg 1 mL 200 mg 25 mg 2 mg 500 mg 50 mg 5 mg
Category	Reagents & Chemicals Biochemicals
Type	Chemicals
Specific against	other
Formula	C15H16ClN3O3
Smiles	ClC1=C(NCCN2CCOCC2)C(=O)c2ncccc2C1=O
ECLASS 10.1	32160000
ECLASS 11.0	32160000
UNSPSC	12000000
Alias	NSC 663284
Shipping Condition	Cool pack
Available
Manufacturer - Targets	Phosphatase\|\|\|Histone Methyltransferase
Shipping Temperature	Cool pack
Storage Conditions	-20°C
Molecular Weight	321, 76
Description	DA-3003-1 (DA-3003-1) is a membrane-permeable, potent and selective Cdc25 dual specificity phosphatase inhibitor with antitumor activity that inhibits Cdc25B2, Cdc25A, Cdc25B2 and Cdc25C.
Pathways	Chromatin/Epigenetic\|\|\|Metabolism
Bioactivity	NSC 663284 is a cell-permeable and irreversible Cdc25 dual specificity phosphatase inhibitor (IC50 for Cdc25B2: 0.21 Î¼M). NSC 663284 inhibits NSD2 (IC50 of 170 nM) through direct interaction with the catalytic SET domain (Kd of 370 nM). NSC 663284 display

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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