GAT211

Item no.	TMO-T27405-5mg
Manufacturer	TargetMol
CASRN	102704-40-5
Amount	5 mg
Quantity options	100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mg 25 mg 500 mg 50 mg 5 mg
Category	Reagents & Chemicals Biochemicals
Type	Chemicals
Specific against	other
Formula	C22H18N2O2
Smiles	[O-][N+](=O)CC(c1c([nH]c2ccccc12)-c1ccccc1)c1ccccc1
ECLASS 10.1	32160000
ECLASS 11.0	32160000
UNSPSC	12000000
Alias	AZ4,GAT-211,AZ 4,GAT 211,AZ-4
Shipping Condition	Cool pack
Available
Manufacturer - Targets	Cannabinoid Receptor\|\|\|cAMP\|\|\|Arrestin
Shipping Temperature	Cool pack
Storage Conditions	-20
Molecular Weight	342.39
Description	GAT211 (AZ-4) is a selective and potent cannabinoid 1 receptor (CB1R) orthosteric modulator (PAM) with high affinity for cAMP and β-arrestin2.GAT211 has IOP-lowering and antipsychotic effects and can be used in the study of epilepsy.
Pathways	GPCR/G Protein
Bioactivity	GAT211 is a CB1 positive allosteric modulator. GAT211 suppresses allodynia and produces synergistic antiallodynic effects with monoacylglycerol lipase and fatty acid amide hydrolase inhibitors in paclitaxel-treated mice.

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Request Data Sheet

Request product datasheet

Request safety datasheet

Simple Order Order Subscription

Amount: 5 mg

available

Compare

Add to wishlist

Get an offer

Request delivery time

Ask a technical question