Comparison

BX795 European Partner

Item no. TMO-T1830-1ml
Manufacturer TargetMol
CASRN 702675-74-9
Amount 1 mL
Quantity options 100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mL 200 mg 25 mg 500 mg 50 mg 5 mg
Category
Type Chemicals
Specific against other
Smiles Ic1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCCNC(=O)c1cccs1
ECLASS 10.1 32160000
ECLASS 11.0 32160000
UNSPSC 12000000
Similar products 702675-74-9
Shipping Condition Cool pack
Available
Manufacturer - Targets
IκB/IKK|||Chk|||PDK|||c-Kit|||CDK|||Autophagy
Shipping Temperature
Cool pack
Storage Conditions
-20
Molecular Weight
591.47
Description
BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity is 140- and 1600-fold for PDK1 over PKA and PKC in cell-free assays, respectively. Meanwhile, the selectivity for PDK1 is 100-fold than GSK3β.
Pathways
NF-κB|||PI3K/Akt/mTOR signaling|||Autophagy|||Cell Cycle/Checkpoint|||Tyrosine Kinase/Adaptors

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 1 mL
Available: In stock
available

Compare

Add to wishlist

Get an offer

Request delivery time

Ask a technical question

Submit a bulk request

Questions about this Product?
 
Close