PFI-1

Item no.	TMO-T6222-2mg
Manufacturer	TargetMol
CASRN	1403764-72-6
Amount	2 mg
Quantity options	100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mL 200 mg 25 mg 2 mg 50 mg 5 mg
Category	Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
Citations	1. Fish PV, et al. J Med Chem, 2012, 55(22), 9831-9837.
Smiles	COc1ccccc1S(=O)(=O)Nc1ccc2NC(=O)N(C)Cc2c1
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Alias	PF-6405761,PFI 1,PFI1
Shipping Condition	Cool pack
Available
Manufacturer - Targets	Apoptosis\|\|\|Epigenetic Reader Domain\|\|\|Autophagy
Shipping Temperature	Cool pack
Storage Conditions	-20
Molecular Weight	347.39
Description	PFI-1 (PF-6405761), a specific BET (bromodomain-containing protein) inhibitor for BRD4, is with the IC50 of 0.22 μM in a cell-free assay.
Pathways	Autophagy\|\|\|Chromatin/Epigenetic\|\|\|Apoptosis
Bioactivity	PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 uM in a cell-free assay.
Receptor	BRD2; BRD4

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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