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Belumosudil

Belumosudil

Item no.	TMO-T6867-10mM
Manufacturer	TargetMol
CASRN	911417-87-3
Amount	1 mL x 10 mM (in DMSO)
Quantity options	100 mg 1 mL x 10 mM (in DMSO) 10 mg 1 mL 25 mg 2 mg 500 mg 50 mg 5 mg
Category	Oncology Reagents & Chemicals Molecules By Organ Hepatic Cancer
Type	Molecules
Specific against	other
Citations	1. Lee JH, et al. Ann Clin Transl Neurol. 2014, 1(1), 2-14.
Smiles	CC(C)NC(=O)COc1cccc(c1)-c1nc(Nc2ccc3[nH]ncc3c2)c2ccccc2n1
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Alias	KD025,Rezurock,ROCK inhibitor,SLx-2119
Shipping Condition	Cool pack
Available
Manufacturer - Targets	ROCK
Shipping Temperature	Cool pack
Storage Conditions	-20
Molecular Weight	452.51
Description	Belumosudil (Rezurock) is an orally available, and specific ROCK2 inhibitor (IC50/Ki: 60/41 nM).
Pathways	Stem Cells\|\|\|Cell Cycle/Checkpoint\|\|\|Cytoskeletal Signaling
Bioactivity	KD025 is an orally available, and selective ROCK2 inhibitor with IC50 and Ki of 60 nM and 41 nM, respectively. Phase 2.
Receptor	ROCK2; ROCK2

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 1 mL x 10 mM (in DMSO)

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